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Cat. No. Product Name Target Signaling Pathways
T2087 AF-353

Ro-4

P2X Receptor Membrane transporter/Ion channel; Neuroscience
AF-353 (Ro-4) 是一种选择性、可口服的 P2X3/P2X2/3 受体拮抗剂,抑制人和大鼠 P2X3 的 pIC50值为 8.0,抑制人 P2X2/3 的 pIC50值为 7.3。
T3559 4-Oxoisotretinoin

Oxoretinoic acid,4-Oxoisotretinoin,Ro 22-6595

Others Others
4-Oxoisotretinoin (Ro 22-6595) 是主要的血液代谢物。
T12745L (4R)-RO5263397

Others Others
(4R)-4-(3-Fluoro-2-methylphenyl)-4,5-dihydro-2-oxazolamin 对 TRACE AMINE ASSOCIATED RECEPTOR (TAAR 1)具有活性,EC50为0.017 μM,可用来研究神经系统疾病。
T8139 Sulfamethoxazole sodium

新诺明钠,Ro 4-2130 sodium,磺胺甲恶唑钠

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Sulfamethoxazole sodium (Ro 4-2130 sodium) 是一种磺胺类抗菌素。它常用于各种尿道病原体的研究,与 Trimethoprim 联用,可用于尿路感染的研究。
T1517 Benserazide hydrochloride

Benserazide HCl,盐酸苄丝肼,Serazide,Ro 4-4602

Dopamine Receptor GPCR/G Protein; Neuroscience
Benserazide hydrochloride (Ro 4-4602) 是一种芳香族 L-氨基酸脱羧酶(AADC)的抑制剂,常用于帕金森病。
T34361 Ro 4-6824

AI3-50843

Ro 4-6824 is a biochemical with immunosuppressive action.
T0885 Sulfamethoxazole

Ro 4-2130,STX 608,磺胺甲恶唑

Antibacterial; Antibiotic; Autophagy Autophagy; Microbiology/Virology
Sulfamethoxazole (STX 608) 是磺胺类抗菌素,用于细菌感染。Sulfonamides 是对氨基苯甲酸的竞争性拮抗剂。
T14489 Azvudine

4-氨基-1-(4-C-叠氮基-2-脱氧-2-氟-BETA-D-呋喃阿拉伯糖基)-2(1H)-嘧啶酮,FNC,RO-0622

HCV Protease; HBV; HIV Protease; Reverse Transcriptase Microbiology/Virology; Proteases/Proteasome
Azvudine (FNC) 是一种有效的核苷逆转录酶抑制剂 (NRTI),对 HIV、HBV 和 HCV 具有抗病毒活性。它抑制耐 NRTI 的病毒株,高效抑制 HIV-1和 HIV-2。
T7745 Diclofensine hydrochloride

4-(3,4-二氯苯)-7-甲氧基-2-甲基-1,2,3,4-四氢异喹啉盐酸盐,Ro 8-4650 hydrochloride

Others; Dopamine Receptor GPCR/G Protein; Neuroscience; Others
Diclofensine hydrochloride (Ro 8-4650 hydrochloride) 是一种高效单胺再摄取抑制剂,在大鼠脑突触体中能够阻断多巴胺 (IC50=0.74 nM)、去甲肾上腺素 (IC50=2.3 nM) 和 5-羟色胺 (IC50=3.7 nM)。
T1488L Procarbazine free base

CB 400-497,NSC-77213,Ro 4-6467/1,Ro 4-6467,Procarbazine

Procarbazine is an antineoplastic chemotherapy drug for the treatment of Hodgkin's lymphoma and certain brain cancers. The drug is metabolized and activated in the liver. It also inhibits MAO thus increasing the effects of sympathomimetics, TCAs, and tyra
T19706 Ro 20-1724

Ro-20-1724,4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone,Ro20-1724

PDE Metabolism
Ro 20-1724 (4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone) 是 cAMP 特异性磷酸二酯酶抑制剂 b>(PDE4/PDE IV),其 Ki=1930 nM,具有神经保护作用。
T13031 Sulfamethoxazole-d4

Ro 4-2130 D4,磺胺甲恶唑 D4

Others Others
Sulfamethoxazole D4 is a deuterium labeled Sulfamethoxazole (Ro 4-2130). Sulfamethoxazole is a sulfonamide bacteriostatic antibiotic.
T11679 Isavuconazole-d4

BAL-4815 D4,RO-0094815 D4,Isavuconazole D4

Others Others
Isavuconazole D4 is a deuterium labeled Isavuconazole. Isavuconazole is a triazole prodrug with antifungal activity against yeasts, molds, and dimorphic fungi.
T12718 RG7800 hydrochloride (1449598-06-4 free base)

RO6885247 hydrochloride,RG7800 hydrochloride

Others Others
RG7800 hydrochloride is an orally active modulator of SMN2 splicing.
T6312 R547

Ro 4584820

Apoptosis; GSK-3; PKA; CDK Apoptosis; Cell Cycle/Checkpoint; PI3K/Akt/mTOR signaling; Stem Cells; Tyrosine Kinase/Adaptors
R547 (Ro 4584820) 是一种口服有效,选择性, ATP 竞争性CDK 抑制剂,对 CDK1/cyclin B、 CDK2/cyclin E 和 CDK4/cyclin D1 作用的Ki 值分别为 2 nM、3 nM、1 nM。
T28595 Ro-0505124

Ro0505124,Ro 0505124

Ro-0505124 is a potent, selective and ATP-competitive inhibitor of cyclin-dependent kinase 4 (CDK4).
T70838 RO27-3225 TFA

RO27-3225, also known as RO273225 is a melanocortin type 4 receptor agonist with EC50 = 1 nM. It may alleviate intestinal dysfuntion and brain damage. It has been investigated for an anti-obesity medication. Ro 27-3225 shows some activity at the MC1 receptor. Ro 27-3225 reverses hemorrhagic shock, reduces multiple organ damage, and improves survival.

化合物

AF-353
Cat.No: T2087
Synonym: Ro-4
Target: P2X Receptor
4-Oxoisotretinoin
Cat.No: T3559
Synonym: Oxoretinoic acid,4-Oxoisotretinoin,Ro 22-6595
Target: Others
(4R)-RO5263397
Cat.No: T12745L
Synonym:
Target: Others
Sulfamethoxazole sodium
Cat.No: T8139
Synonym: 新诺明钠,Ro 4-2130 sodium,磺胺甲恶唑钠
Target: Others, Antibacterial, Antibiotic
Benserazide hydrochloride
Cat.No: T1517
Synonym: Benserazide HCl,盐酸苄丝肼,Serazide,Ro 4-4602
Target: Dopamine Receptor
Ro 4-6824
Cat.No: T34361
Synonym: AI3-50843
Target:
Sulfamethoxazole
Cat.No: T0885
Synonym: Ro 4-2130,STX 608,磺胺甲恶唑
Target: Antibacterial, Antibiotic, Autophagy
Azvudine
Cat.No: T14489
Synonym: 4-氨基-1-(4-C-叠氮基-2-脱氧-2-氟-BETA-D-呋喃阿拉伯糖基)-2(1H)-嘧啶酮,FNC,RO-0622
Target: HCV Protease, HBV, HIV Protease, Reverse Transcriptase
Diclofensine hydrochloride
Cat.No: T7745
Synonym: 4-(3,4-二氯苯)-7-甲氧基-2-甲基-1,2,3,4-四氢异喹啉盐酸盐,Ro 8-4650 hydrochloride
Target: Others, Dopamine Receptor
Procarbazine free base
Cat.No: T1488L
Synonym: CB 400-497,NSC-77213,Ro 4-6467/1,Ro 4-6467,Procarbazine
Target:
Ro 20-1724
Cat.No: T19706
Synonym: Ro-20-1724,4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone,Ro20-1724
Target: PDE
Sulfamethoxazole-d4
Cat.No: T13031
Synonym: Ro 4-2130 D4,磺胺甲恶唑 D4
Target: Others
Isavuconazole-d4
Cat.No: T11679
Synonym: BAL-4815 D4,RO-0094815 D4,Isavuconazole D4
Target: Others
RG7800 hydrochloride (1449598-06-4 free base)
Cat.No: T12718
Synonym: RO6885247 hydrochloride,RG7800 hydrochloride
Target: Others
R547
Cat.No: T6312
Synonym: Ro 4584820
Target: Apoptosis, GSK-3, PKA, CDK
Ro-0505124
Cat.No: T28595
Synonym: Ro0505124,Ro 0505124
Target:
RO27-3225 TFA
Cat.No: T70838
Synonym:
Target:
TargetMol Loading
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